Table of medication secreted in kidney

This is a table of medications that are secreted in the kidney.

Acid medication are, because of pH partition, secreted to a higher extent when urine is basic. In the same way, basic medications are secreted to a higher extent when urine is acidic.

Medication Location Acid or base anion or cation Percentage excreted
para-aminohippurate proximal tubuleAcidanion
furosemide proximal tubuleAcidanion100-75
glucuronic acid-conjugates proximal tubuleAcid
glycine conjugates proximal tubuleAcid
indometacin proximal tubuleAcidanion
methotrexate proximal tubuleAcid100-75
penicillin proximal tubuleAcidanion75-50
(benzylpenicillin)
probenecid proximal tubuleAcidanion
sulphate conjugates proximal tubuleAcid
thiazide diuretics proximal tubuleAcid
uric acid proximal tubuleAcid
amiloride proximal tubuleBasecation
dopamine proximal tubuleBase
histamine proximal tubuleBase
mepacrine proximal tubuleBase
morphine proximal tubuleBasecation
pethidine proximal tubuleBase
quaternary ammonium compounds proximal tubuleBase
quinine proximal tubuleBasecation
5-hydroxytryptamine (serotonin) proximal tubuleBase
triamterene proximal tubuleBase
gentamicin 100-75
atenolol 100-75
digoxin 100-75
cimetidine cation75-50
tetracycline 75-50
(oxytetracycline)
neostigmine 75-50
propantheline ~50
tubocurarine ~50
acetazolamide proximal tubuleanion
chlorothiazide proximal tubuleanion
saccharin proximal tubuleanion
salicylate proximal tubuleanion
atropine proximal tubulecation
NMN proximal tubulecation
paraquat proximal tubulecation
procainamide proximal tubulecation
tetraethylammonium proximal tubulecation
chlorpromazine proximal tubulecation
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